An Activity-Based Probe for Cathepsin K Imaging with Excellent Potency and Selectivity
| Document Type: | Article |
|---|---|
| Language: | English |
| Author: | Carina Lemke, Jakub Benýšek, Dominik Brajtenbach, Christian Breuer, Adéla Jílková, Martin Horn, Michal Buša, Lenka Ulrychová, Annika Illies, Katharina F. Kubatzky, Ulrike Bartz, Michael Mareš, Michael Gütschow |
| Parent Title (English): | Journal of Medicinal Chemistry |
| Volume: | 64 |
| Issue: | 18 |
| First Page: | 13793 |
| Last Page: | 13806 |
| ISSN: | 0022-2623 |
| DOI: | https://doi.org/10.1021/acs.jmedchem.1c01178 |
| PMID: | https://pubmed.ncbi.nlm.nih.gov/34473502 |
| Publisher: | American Chemical Society (ACS) |
| Date of first publication: | 2021/09/02 |
| Copyright: | © 2021 American Chemical Society |
| Funding: | C.L. thanks the Bonn International Graduate School of Drug Sciences (BIGS-DrugS)/BMBF for obtaining a grant (16GW0025). C.B. was supported by a grant from the Department of Natural Sciences, University of Applied Sciences Bonn-Rhein-Sieg. M.M., J.B., A.J., M.H., M.B., and L.U. were supported by the project ChemBioDrug CZ.02.1.01/0.0/0.0/16_019/0000729 from ERDF/OPRDE, Gilead Sciences & IOCB Research Center, and the institutional project RVO 61388963. |
| Departments, institutes and facilities: | Fachbereich Angewandte Naturwissenschaften |
| Dewey Decimal Classification (DDC): | 5 Naturwissenschaften und Mathematik / 54 Chemie / 540 Chemie und zugeordnete Wissenschaften |
| Entry in this database: | 2021/09/06 |
